Yangonin
http://dbpedia.org/resource/Yangonin an entity of type: Thing
ヤンゴニン (Yangonin) は、カヴァに含まれる6つの主なカヴァラクトンのうちの1つである。に対する結合親和性 (Ki = 0.72 μM )を持ち、アゴニストとして作用する。
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Yangonin is one of the six major kavalactones found in the kava plant. It has been shown to possess binding affinity for the cannabinoid receptor CB1 (Ki = 0.72 μM), and selectivity vs. the CB2 receptor (Ki >10 μM) where it behaves as an agonist. The CB1 receptor affinity of yangonin suggests that the endocannabinoid system might contribute to the complex human psychopharmacology of the traditional kava drink and the anxiolytic preparations obtained from the kava plant.
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ヤンゴニン
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Yangonin
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24225422
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1099982923
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Yangonin.svg
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Yangonin02.png
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200
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4
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changed
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412605522
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Yangonin is one of the six major kavalactones found in the kava plant. It has been shown to possess binding affinity for the cannabinoid receptor CB1 (Ki = 0.72 μM), and selectivity vs. the CB2 receptor (Ki >10 μM) where it behaves as an agonist. The CB1 receptor affinity of yangonin suggests that the endocannabinoid system might contribute to the complex human psychopharmacology of the traditional kava drink and the anxiolytic preparations obtained from the kava plant. Further in vitro studies have also demonstrated yangonin to be an inhibitor of monoamine oxidase, with a moderate preference for isozyme B, which could open the door to a wide range of interactions.
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ヤンゴニン (Yangonin) は、カヴァに含まれる6つの主なカヴァラクトンのうちの1つである。に対する結合親和性 (Ki = 0.72 μM )を持ち、アゴニストとして作用する。
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4123
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4-Methoxy-6-[(E)-2-(4-methoxyphenyl)ethen-1-yl]-2H-pyran-2-one
