4-Fluorophenibut
http://dbpedia.org/resource/4-Fluorophenibut an entity of type: Thing
4-氨基-3-(4-氟苯基)丁酸或β-氨基甲基-4-氟苯丙酸（研发代号CGP-11130）是一种有机化合物，化学式为C10H12FNO2。它是GABAB受体激动剂，但从未上市。它可由4-硝基-3-(4-氟苯基)丁醛经氧化至羧酸，再由硼氢化钠还原硝基，调节pH至3~4得到。 立陶宛 和匈牙利的法律将其禁售。
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4-Fluorophenibut (developmental code name CGP-11130; also known as β-(4-fluorophenyl)-γ-aminobutyric acid or β-(4-fluorophenyl)-GABA) is a GABAB receptor agonist which was never marketed. It is selective for the GABAB receptor over the GABAA receptor (IC50 = 1.70 μM and > 100 μM, respectively). The drug is a GABA analogue and is closely related to baclofen (β-(4-chlorophenyl)-GABA), tolibut (β-(4-methylphenyl)-GABA), and phenibut (β-phenyl-GABA). It is less potent as a GABAB receptor agonist than baclofen but more potent than phenibut.
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4-Fluorophenibut
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4-氨基-3-(4-氟苯基)丁酸
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CGP-11130; β--γ-aminobutyric acid; β--GABA; Baflofen; Fluorophenibut; F-Phenibut; Fluoribut
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6
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4-Fluorophenibut (developmental code name CGP-11130; also known as β-(4-fluorophenyl)-γ-aminobutyric acid or β-(4-fluorophenyl)-GABA) is a GABAB receptor agonist which was never marketed. It is selective for the GABAB receptor over the GABAA receptor (IC50 = 1.70 μM and > 100 μM, respectively). The drug is a GABA analogue and is closely related to baclofen (β-(4-chlorophenyl)-GABA), tolibut (β-(4-methylphenyl)-GABA), and phenibut (β-phenyl-GABA). It is less potent as a GABAB receptor agonist than baclofen but more potent than phenibut. The substance is sometimes referred to as 4F-phenibut or F-phenibut and colloquially as fluorobut.
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4-氨基-3-(4-氟苯基)丁酸或β-氨基甲基-4-氟苯丙酸（研发代号CGP-11130）是一种有机化合物，化学式为C10H12FNO2。它是GABAB受体激动剂，但从未上市。它可由4-硝基-3-(4-氟苯基)丁醛经氧化至羧酸，再由硼氢化钠还原硝基，调节pH至3~4得到。 立陶宛 和匈牙利的法律将其禁售。
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3539
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